Products & Services
Ready-to-use ADME assay kits with built in quality control.
TRANSIL Plasma Protein Binding Assays
Assessing plasma protein binding is important because only the unbound fraction (fu) of a drug can penetrate cell membranes. Thus, only a drug’s ...
-
TRANSIL HSA Binding Kit
Determination of Drug-Albumin Binding Constants for Prediction of Plasma Protein Binding The TRANSIL HSA Binding Kit determines the binding affinity...Regular price From €534.00Regular priceUnit price / perSale price From €534.00 -
TRANSIL AGP Binding Kit
Determination of Drug–α1-Acid Glycoprotein Binding Constants for Characterizing Plasma Protein Binding The TRANSIL AGP Binding Kit determines the binding affinity...Regular price €1,055.00Regular priceUnit price / perSale price €1,055.00 -
TRANSIL PPB Binding Kit
Rapid Determination of Human Plasma Protein Binding Using Immobilized Albumin and AGP The TRANSIL PPB Binding Kit enables rapid determination...Regular price €688.00Regular priceUnit price / perSale price €688.00 -
TRANSIL RSA Binding Kit
Determination of Drug–Rat Albumin Binding Constants for Preclinical Pharmacokinetic Studies The TRANSIL RSA Binding Kit enables mechanistic characterization of drug...Regular price €1,364.00Regular priceUnit price / perSale price €1,364.00 -
TRANSIL MSA Binding Kit
Determination of Drug–Mouse Albumin Binding Constants for Interpretation of Mouse Pharmacokinetic Studies The TRANSIL MSA Binding Kit enables mechanistic characterization...Regular price €1,984.00Regular priceUnit price / perSale price €1,984.00 -
TRANSIL High Sensitivity Binding Kit
When Conventional Plasma Protein Binding Assays Fail Measure the unbound fraction of compounds with fu < 1%, strong non-specific binding,...Regular price From €471.50Regular priceUnit price / perSale price From €471.50
TRANSIL Membrane Binding & Permeability Assays
Drug transport can broadly be divided into transcellular and paracellular processes. Transcellular movement, which involves the passage of drugs ...
-
TRANSIL Brain Absorption Kit
Predict Brain Exposure Early in Drug Discovery The TRANSIL Brain Absorption Kit enables rapid in-vitro prediction of brain tissue binding,...Regular price From €714.00Regular priceUnit price / perSale price From €714.00 -
TRANSIL Intestinal Absorption Kit
Predict Intestinal Permeability from Direct Membrane Interaction The TRANSIL Intestinal Absorption Kit directly measures drug affinity to phospholipid membranes and...Regular price From €533.50Regular priceUnit price / perSale price From €533.50 -
TRANSIL Metabolic Bias Kit
Correct Metabolic Rate Bias in Microsomal and Hepatocyte Stability Assays Rapid measurement of membrane binding to calculate fu(mic) and fu(hepatocyte)...Regular price €651.00Regular priceUnit price / perSale price €651.00 -
TRANSIL Membrane Affinity Kit
Measure Membrane Affinity – The Mechanistic Alternative to LogP Rapid determination of compound–membrane interaction in a cell-free system. Use as...Regular price From €534.00Regular priceUnit price / perSale price From €534.00 -
TRANSIL Intracellular Binding Kit
Predict Intracellular Drug Binding from Phospholipid Affinity Estimate intracellular unbound drug fractions (fu,cell) in minutes using a rapid cell- free...Regular price From €909.00Regular priceUnit price / perSale price From €909.00
Assay Development & Consulting
Assessing plasma protein binding is important because only the unbound fraction (fu) of a drug can penetrate cell membranes.